BindingDB PrimarySearch

Found 35 for UniProtKB: Q64133

Amine oxidase [flavin-containing] A(Mus musculus)
University of Cambridge

Curated by ChEMBL

BDBM50148573((E,E)-1-piperoylpiperidine | 1-[(2E,4E)-5-(1,3-ben...)copy SMILEScopy InChI

Ki: 1.90E+4nMAssay Description:Inhibition of mouse brain MAOAMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2000264PubMed

Amine oxidase [flavin-containing] A(Mus musculus)
University of Cambridge

Curated by ChEMBL

BDBM50305644((2E,4E)-5-Benzo[1,3]dioxol-5-yl-penta-2,4-dienoic ...)copy SMILEScopy InChI

Ki: 2.71E+4nMAssay Description:Inhibition of mouse brain MAOAMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2000264PubMed

Amine oxidase [flavin-containing] A(Mus musculus)
University of Cambridge

Curated by ChEMBL

BDBM50490813(CHEMBL2346911)copy SMILEScopy InChI

IC50: 0.00100nMAssay Description:Inhibition of mouse brain MAO-AMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q25T3PCSPubMed

Amine oxidase [flavin-containing] A(Mus musculus)
University of Cambridge

Curated by ChEMBL

BDBM50361373(AURAPTENE)copy SMILEScopy InChI

IC50: 0.0350nMAssay Description:Inhibition of mouse brain MAO-AMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q25T3PCSPubMed

Amine oxidase [flavin-containing] A(Mus musculus)
University of Cambridge

Curated by ChEMBL

BDBM50586985(CHEMBL5082735)copy SMILES

IC50: 7.80nMAssay Description:Displacement of [18F]-FEH from MAO-A in mouse brain homogenate incubated for 60 mins by imaging analysisMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2PC3698PubMed

Amine oxidase [flavin-containing] A(Mus musculus)
University of Cambridge

Curated by ChEMBL

BDBM50586984(CHEMBL5084771)copy SMILES

IC50: 51nMAssay Description:Displacement of [18F]-FEH from MAO-A in mouse brain homogenate incubated for 60 mins by imaging analysisMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2PC3698PubMed

Amine oxidase [flavin-containing] A(Mus musculus)
University of Cambridge

Curated by ChEMBL

BDBM50586986(CHEMBL5091624)copy SMILES

IC50: 1.00E+3nMAssay Description:Displacement of [18F]-FEH from MAO-A in mouse brain homogenate incubated for 60 mins by imaging analysisMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2PC3698PubMed

Amine oxidase [flavin-containing] A(Mus musculus)
University of Cambridge

Curated by ChEMBL

BDBM50586977(CHEMBL5081957)copy SMILES

IC50: 1.00E+3nMAssay Description:Displacement of [18F]-FEH from MAO-A in mouse brain homogenate incubated for 60 mins by imaging analysisMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2PC3698PubMed

Amine oxidase [flavin-containing] A(Mus musculus)
University of Cambridge

Curated by ChEMBL

BDBM50586972(CHEMBL5088921)copy SMILES

IC50: 1.00E+3nMAssay Description:Displacement of [18F]-FEH from MAO-A in mouse brain homogenate incubated for 60 mins by imaging analysisMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2PC3698PubMed

Amine oxidase [flavin-containing] A(Mus musculus)
University of Cambridge

Curated by ChEMBL

BDBM50586973(CHEMBL5077904)copy SMILES

IC50: 1.00E+3nMAssay Description:Displacement of [18F]-FEH from MAO-A in mouse brain homogenate incubated for 60 mins by imaging analysisMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2PC3698PubMed

Amine oxidase [flavin-containing] A(Mus musculus)
University of Cambridge

Curated by ChEMBL

BDBM50586974(CHEMBL5090407)copy SMILES

IC50: 1.00E+3nMAssay Description:Displacement of [18F]-FEH from MAO-A in mouse brain homogenate incubated for 60 mins by imaging analysisMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2PC3698PubMed

Amine oxidase [flavin-containing] A(Mus musculus)
University of Cambridge

Curated by ChEMBL

BDBM50586975(CHEMBL5081662)copy SMILES

IC50: 1.00E+3nMAssay Description:Displacement of [18F]-FEH from MAO-A in mouse brain homogenate incubated for 60 mins by imaging analysisMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2PC3698PubMed

Amine oxidase [flavin-containing] A(Mus musculus)
University of Cambridge

Curated by ChEMBL

BDBM50586976(CHEMBL5092563)copy SMILES

IC50: 1.00E+3nMAssay Description:Displacement of [18F]-FEH from MAO-A in mouse brain homogenate incubated for 60 mins by imaging analysisMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2PC3698PubMed

Amine oxidase [flavin-containing] A/B(Mus musculus)
Fudan University

Curated by ChEMBL

BDBM50523994(CHEMBL461985)copy SMILEScopy InChI

IC50: 1.06E+3nMAssay Description:Inhibition of mouse brain monoamine oxidaseMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2BG2SD6PubMed

Amine oxidase [flavin-containing] A(Mus musculus)
University of Cambridge

Curated by ChEMBL

BDBM50531888(CHEMBL4162879)copy SMILEScopy InChI

IC50: 1.30E+3nMAssay Description:Inhibition of MAO-A in mouse brain mitochondrial fraction using kynuramine as substrate after 30 mins by fluorometric analysisMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2WW7N5DPubMed

Amine oxidase [flavin-containing] A(Mus musculus)
University of Cambridge

Curated by ChEMBL

BDBM50491068(Lacinartin)copy SMILEScopy InChI

IC50: 5.70E+3nMAssay Description:Inhibition of MAO-A in mouse brain mitochondrial fraction using kynuramine as substrate by fluorometric analysisMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2WW7N5DPubMed

Amine oxidase [flavin-containing] A(Mus musculus)
University of Cambridge

Curated by ChEMBL

BDBM50491068(Lacinartin)copy SMILEScopy InChI

IC50: 5.70E+3nMAssay Description:Inhibition of mouse brain MAO-AMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q25T3PCSPubMed

Amine oxidase [flavin-containing] A(Mus musculus)
University of Cambridge

Curated by ChEMBL

BDBM50084137(2-Methyl-6-(phenylethynyl)pyridine | 2-Methyl-6-ph...)copy SMILEScopy InChI

IC50: 8.00E+3nMAssay Description:Tested for in vitro antagonistic activity against Monoamine oxidaseMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q28P5ZT7PubMed

Amine oxidase [flavin-containing] A(Mus musculus)
University of Cambridge

Curated by ChEMBL

BDBM50021398(CHEBI:18088 | FORMONONETIN | NSC-93360)copy SMILEScopy InChI

IC50: 2.12E+4nMAssay Description:Inhibition of mouse MAO-A preincubated for 15 mins followed by addition of kynuramine as substrate measured after 30 mins by fluorometric analysisMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2M90D5HPubMed

Amine oxidase [flavin-containing] A(Mus musculus)
University of Cambridge

Curated by ChEMBL

BDBM50122758(2-methyl-4-(pyridin-3-ylethynyl)thiazole | 3-(2-(2...)copy SMILEScopy InChI

IC50: 3.00E+4nMAssay Description:Tested for in vitro antagonistic activity against Monoamine oxidase AMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q28P5ZT7PubMed

Amine oxidase [flavin-containing] A(Mus musculus)
University of Cambridge

Curated by ChEMBL

BDBM50017857(3-(3,4-Dihydroxy-5-nitro-phenyl)-1-phenyl-propenon...)copy SMILEScopy InChI

IC50: 5.00E+4nMAssay Description:Inhibitory activity against the Monoamine oxidase AMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2GF0SHPPubMed

Amine oxidase [flavin-containing] A(Mus musculus)
University of Cambridge

Curated by ChEMBL

BDBM50017850(1-(3,4-Dihydroxy-phenyl)-2-methyl-propan-1-one | C...)copy SMILEScopy InChI

IC50: 5.00E+4nMAssay Description:Inhibitory activity against the Monoamine oxidase AMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2GF0SHPPubMed

Amine oxidase [flavin-containing] A(Mus musculus)
University of Cambridge

Curated by ChEMBL

BDBM50017845(3-(3,4-Dihydroxy-5-nitro-phenyl)-1-(3,4,5-trimetho...)copy SMILEScopy InChI

IC50: 5.00E+4nMAssay Description:Inhibitory activity against the Monoamine oxidase AMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2GF0SHPPubMed

Amine oxidase [flavin-containing] A(Mus musculus)
University of Cambridge

Curated by ChEMBL

BDBM50193718(2-(2,4-dihydroxy-phenyl)-5-hydroxy-8,8-dimethyl-3-...)copy SMILEScopy InChI

IC50: 8.00E+4nMAssay Description:Inhibition at monoamine oxidase in mouse brainMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2K938CCPubMed

Amine oxidase [flavin-containing] A(Mus musculus)
University of Cambridge

Curated by ChEMBL

BDBM50175016(1,3,6,7-tetrahydroxy-4-(1,1-dimethyl-2-propenyl)-8...)copy SMILEScopy InChI

IC50: 8.83E+4nMAssay Description:Inhibition at monoamine oxidase in mouse brainMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2K938CCPubMed

Amine oxidase [flavin-containing] A(Mus musculus)
University of Cambridge

Curated by ChEMBL

BDBM50193719((S)-5,7,7'-trihydroxy-2',2'-dimethyl-6-(3-methylbu...)copy SMILEScopy InChI

IC50: 8.97E+4nMAssay Description:Inhibition at monoamine oxidase in mouse brainMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2K938CCPubMed

Amine oxidase [flavin-containing] A(Mus musculus)
University of Cambridge

Curated by ChEMBL

BDBM50593239(CHEBI:5637 | CHEMBL12367 | EN300-17866)copy SMILES

IC50: 1.00E+5nMMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2H70KTGPubMed

Amine oxidase [flavin-containing] A(Mus musculus)
University of Cambridge

Curated by ChEMBL

BDBM50175017(3,6,8-trihydroxy-2-methoxy-1-(3-methylbut-2-enyl)-...)copy SMILEScopy InChI

IC50: 1.50E+5nMAssay Description:Inhibition at monoamine oxidase in mouse brainMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2K938CCPubMed

Amine oxidase [flavin-containing] A(Mus musculus)
University of Cambridge

Curated by ChEMBL

BDBM50217269(1,3,6,7-tetrahydroxy-4-(1,1-dimethylallyl)-8-(3-hy...)copy SMILEScopy InChI

IC50: 1.50E+5nMAssay Description:Inhibition at monoamine oxidase in mouse brainMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2K938CCPubMed

Amine oxidase [flavin-containing] A(Mus musculus)
University of Cambridge

Curated by ChEMBL

BDBM50217268(1,6,7-trihydroxy-3-methoxy-2,4-(3-methylbut-2-enyl...)copy SMILEScopy InChI

IC50: 1.50E+5nMAssay Description:Inhibition at monoamine oxidase in mouse brainMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2K938CCPubMed

Amine oxidase [flavin-containing] A(Mus musculus)
University of Cambridge

Curated by ChEMBL

BDBM50217272(1,6,7-trihydroxy-8-(3-methylbut-2-enyl)-4',5'-dihy...)copy SMILEScopy InChI

IC50: 1.50E+5nMAssay Description:Inhibition at monoamine oxidase in mouse brainMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2K938CCPubMed

Amine oxidase [flavin-containing] A(Mus musculus)
University of Cambridge

Curated by ChEMBL

BDBM50217273(CHEMBL390040 | isocudraxanthone K)copy SMILEScopy InChI

IC50: 1.50E+5nMAssay Description:Inhibition at monoamine oxidase in mouse brainMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2K938CCPubMed

Amine oxidase [flavin-containing] A(Mus musculus)
University of Cambridge

Curated by ChEMBL

BDBM50217274((-)-Cudraflavone A | 3,8-Dihydroxy-11,11-dimethyl-...)copy SMILEScopy InChI

IC50: 1.50E+5nMAssay Description:Inhibition at monoamine oxidase in mouse brainMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2K938CCPubMed

Amine oxidase [flavin-containing] A(Mus musculus)
University of Cambridge

Curated by ChEMBL

BDBM50175013(1,3,6,7-tetrahydroxy-5-(3-methylbut-2-enyl)-2-(2-m...)copy SMILEScopy InChI

IC50: 1.50E+5nMAssay Description:Inhibition at monoamine oxidase in mouse brainMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2K938CCPubMed

Amine oxidase [flavin-containing] A(Mus musculus)
University of Cambridge

Curated by ChEMBL

BDBM50217270(1,3,6,7-tetrahydroxy-4-(1,1-dimethylallyl)xanthone...)copy SMILEScopy InChI

IC50: 1.50E+5nMAssay Description:Inhibition at monoamine oxidase in mouse brainMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2K938CCPubMed

Targets 2 ▿
- Amine oxidase [flavin-containing] A 34
- Amine oxidase [flavin-containing] A/B 1
Publications 8 ▿
- J Nat Prod 70: 1207-9 (2007) 11
- Bioorg Med Chem 21: 2434-50 (2013) 3
- J Med Chem 32: 841-6 (1989) 3
- Bioorg Med Chem Lett 29: 839-843 (2019) 2
- Bioorg Med Chem Lett 20: 537-40 (2010) 2
- J Med Chem 46: 204-6 (2003) 2
- Bioorg Med Chem 27: 2027-2040 (2019) 1
- Bioorg Med Chem Lett 26: 4714-4719 (2016) 1
Institutions 7 ▿
- [Chungbuk National University] 11
- [Orion Corporation Ltd., R.C. Patel Institute of Pharmaceutical Education and Research, Sunchon National University] 3
- [Orion Corporation Ltd., R.C. Patel Institute of Pharmaceutical Education and Research, Sunchon National University] 3
- [Orion Corporation Ltd., R.C. Patel Institute of Pharmaceutical Education and Research, Sunchon National University] 3
- [Merck Research Laboratories, University of Cambridge] 2
- [Merck Research Laboratories, University of Cambridge] 2
- [Fudan University] 1
Affinity: 0.0010 to 1.5E+5 nM▿
- Ki 2
- IC50 33
- Affinity ≤ nM
Xtal structures: 0
Docked structures: 0
Catalog Cmpds: 12